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Antidepressant "Velaksin": haƙuri shedu, umarnin don amfani, analogs

Zan iya sayan antidepressants ba tare da takardar sayen magani? A jerin irin kayayyakin ba manyan. Wannan shi ne saboda cewa su iya zama jaraba, da kuma rundunar illa. Saboda haka, kafin shan irin wannan hanyar, a tabbatar ziyarci wani gwani.

janar bayanai

Mawuyacin ba a bi ta da kwayoyi. Amma don inganta aiki na juyayi tsarin, da yawa likitoci har yanzu rubũta zuwa ga marasa lafiya daban-daban antidepressants. Daya daga cikinsu shi ne magani "Velaksin". Shedu game da wannan kayan aiki da kuma ta siffofin da umarnin don amfani za a gabatar a kasa.

A abun da ke ciki na miyagun ƙwayoyi, ta hanyar samar da

A abin da fom da shi na samar da wani antidepressant matsayin "Velaksin"? Allunan, kuma ya capsules - ne kawai siffofin da miyagun ƙwayoyi.

Allunan "Velaksin" ne fari, kwarzana a gefe daya "E741", da kuma wani madauwari lebur siffar da chamfer. Su aiki sashi ne venlafaxine, wanda aka wakilta a cikin wani nau'i na hydrochloride. Har ila yau, a hada a cikin wannan magani hada da karin gyara irin yadda colloidal silica anhydrous, lactose monohydrate, sodium sitaci glycolate, magnesium stearate da Hukumar ta MCC.

Cushe Allunan a bororo fakitoci kuma cartons bi da bi.

Drug "Velaksin" - capsules, umarnin don amfani da ake kewaye a cikin marufi, takarda, gelatin da kuma m. Suna da orange-kasa-kasa hula da kuma wani colorless substrate. The aiki bangaren na wannan nau'i ne ma a fili venlafaxine. Bugu da kari to abun da ke ciki na wannan magani hada da ƙarin sinadaran.

Kamar yadda miyagun ƙwayoyi ayyuka?

"Velaksin" - wani sabon ƙarni na anti-depressant. Bisa ga sinadaran tsarin na aiki abu ba ya kamãta da kõwa da aka sani aji na antidepressants (msl, tricyclic, tetracyclic, ko wasu). Masana sun ce cewa da miyagun ƙwayoyi ne aiki enantiomer 2 racemate.

A manufa na mataki na wannan magani aka alaka da ikon potentiate da CNS jijiya turu watsa.

Bisa ga umarnin, venlafaxine da manyan metabolite (EFA ko O-desmetilvenlafaksin) wakiltar m hanawa na reuptake na norepinephrine da serotonin da kuma raunana hanawa na dopamine reuptake. Ba za mu iya ce cewa wadannan abubuwa suna iya rage beta-adrenergic aiki bayan wani guda kuma m magani. EFA da venlafaxine ne daidai da tasiri da reuptake na neurotransmitters.

Abin da kuma ne na ƙwarai miyagun ƙwayoyi "Velaksin"? Guide rahoton cewa aiki sashi daga cikin miyagun ƙwayoyi yana da wani dangantaka da n- da m-cholinergic rabe, kwakwalwa α1-adrenoceptors da histamine H1-rabe. Bugu da ƙari, shi damuarn da mataki na Mao, kuma yana da babu kama da fentsiklidinovymi, opioid, benzodiazepine da NMDA-rabe.

A motsi da miyagun ƙwayoyi

ko da miyagun ƙwayoyi ne tunawa, "Velaksin" (Allunan)? Umurnai na Amfani furta cewa aiki bangaren na wannan magani yana da kyau quite tunawa daga gut. Bayan guda kashi na medicament a wani sashi na 25-150 MG na ta cincirindo a jini da aka kai bayan 2.4 hours. Kamar wancan venlafaxine aka baje metabolized lokacin farko da izinin tafiya a cikin hanta. Idan da miyagun ƙwayoyi ne riƙi da abinci, yayin da ta ganiya taro ƙaruwa ta 27-30 minti a cikin jini.

Babban metabolite aka dauke a wajen O-desmetilvenlafaksin. Its rabin rayuwa da kuma kawar rabin-rai na venlafaxine ne 11 da kuma 5 hours, bi da bi (fitarwa a canzawa form ta kodan).

A motsi da kwayoyi a cikin musamman na asibiti yanayi

Drug "Velaksin" wa'azi ake bukata karatu a mutane da cirrhosis na hanta yana da sauran sanadin motsi fasali. jini taro na miyagun ƙwayoyi ya karu a cikin wadannan marasa lafiya, da kuma ta kudi na tukar tumbi, a akasin haka, rage.

A tsanani na koda insufficiency, koda gazawar da kuma matsakaici total yarda EFA da venlafaxine an rage da kuma kawar rabin-rai lokaci ne tsawo.

Ya kamata kuma a lura da cewa, jinsi da shekaru na haƙuri ba zai tasiri a pharmacokinetics da miyagun ƙwayoyi a karkashin shawara.

alamomi ga

Me ya sa muke bukatar wani kayan aiki irin su "Velaksin"? A amfani da wannan magani aka nuna a cikin ciki na daban-daban asalin (domin lura da prophylaxis).

Haramta da nada

A karkashin abin da yanayi ba zai iya yin amfani da miyagun ƙwayoyi "Velaksin"? Reviews da marasa lafiya da likitoci da'awar cewa wannan magani ne contraindicated zuwa sama:

  • yayin da samun Mao hanawa .
  • a mai tsanani koda cuta.
  • a lokacin da wani da ake zargin ko kafa ciki.
  • a cikin tsanani da cuta da hanta.
  • a lokacin shayarwa.
  • a samartaka da yara, da cewa shi ne, har da shekaru masu rinjaye.
  • tare da babban ji na ƙwarai to miyagun ƙwayoyi.

Bugu da ƙari, wannan magani ya kamata a hankali dauka a m angina, tsokar zuciya infarction (ciki har da sabon hijira), hauhawar jini, convulsions tarihi, tachycardia, nauyi asara, ta ƙara intraocular matsa lamba, kwana-ƙulli glaucoma, predisposition zuwa zub da jini daga mucous da kuma fata, manic jihohi.

Drug "Velaksin" (Allunan): umarnin don amfani da

Antidepressant "Velaksin" Ya kamata a dauki kawai a lokacin da wani abinci. The shawarar farawa kashi na da miyagun ƙwayoyi ne 75 MG, ya raba a 2 raba allurai (Ina nufin, 37.5 MG sau biyu a rana), a kowace rana.

Idan bayan makonni da dama na far, haƙuri da yanayin da ya ba inganta, da kullum kashi ne ya karu zuwa 150 MG a rana, a biyu raba allurai (Ina nufin, 75 MG sau biyu a rana).

Idan haƙuri bukatar hakan kashi na wani antidepressant (msl, manyan depressive cuta, ko wasu yanayi bukata far tsit), sa'an nan da m iya designate 150 MG na miyagun ƙwayoyi a 2 hours, sa'an nan a hankali kara da kashi da 75 MG (2-3 kwanaki daga baya) to cimma da ake so sakamakon.

Bisa ga umarnin, matsakaicin sashi "Velaksina" ne 375 MG da rana. Bayan cimma da ake so sakamako, shi za a iya hankali saukar zuwa m matakin.

Da komowa yin rigakafi da goyon baya far

Taimaka kula da kudi na iya daukar daga watanni shida. A wannan yanayin, da magani dauka a kadan allurai.

A m koda insufficiency gyara dosing regimen ake bukata. A irin wannan cuta matsakaici kashi shawarar ƙananan ta 25-50%. Ya kamata kuma a lura da cewa venlafaxine kamata ba a yi amfani a cikin tsanani na koda insufficiency, tun ba bayani a kan aminci da irin wannan far zuwa ranar, ba.

Mutanen da suke kan hemodialysis, ya sami 50% daga cikin saba kullum sashi daga cikin miyagun ƙwayoyi bayan da zaman iyakar.

Domin m hanta insufficiency gyara dosing regimen ne ma ba bukata. Lokacin da cuta ne matsakaici kashi ya kamata a rage by 50%. Game da m hanta gazawar, a wannan yanayin da yin amfani da venlafaxine da aka haramta.

A cikin tsofaffi, da miyagun ƙwayoyi "Velaksin" ya kamata a yi amfani da tare da matsananci hankali. Wannan shi ne saboda da yiwu take hakkin da kodan. A marasa lafiya dole ne rubũta mafi ƙasƙanci tasiri kashi. A wannan yanayin, da mãsu haƙuri ya zama karkashin m likita dubawa.

soke antidepressant

Bayan kammala na karbar magani ya kamata a dauke su rage kashi hankali (a cikin mako guda). Yana ake bukata don tsayar da yanayin haƙuri, domin rage girman hadarin m halayen hade da yarjejeniyoyin da miyagun ƙwayoyi.

A lokacin da ake bukata domin cikakken lõkacin fatara daga cikin magani, ya dogara a kan sashi, duration na far da mutum zuwa mutum.

illa

Mene ne maras so effects da miyagun ƙwayoyi zai iya sa "Velaksin"? Shedu ce cewa ci gaban da wadanda ko wasu m events wadannan da yin amfani da wannan kayan aiki ya dogara da kashi samu.

A mafi m halayen bayyana korau hali hada da wadannan:

  • hauhawar jini, rage ci, mahaukaci mafarkai, maƙarƙashiya, rashin barci, tashin zuciya, flushing na fata, tremors, amai, tsoka cramps, bushe baki.
  • hallucinations, hepatitis, nauyi asara, tachycardia, hyponatremia, apathy, postural hypotension, juwa ko jiri, manic dauki, m excitability, yawning, paresthesia, neuroleptic ciwo, mãyen, serotonergic ciwo.
  • ya karu tsoka sautin, seizures, dysuria, photosensitivity, urinary riƙewa, anorgasmia.
  • zub da jini a cikin fata, mahaukaci kawowa, menorrhagia, rage libido, sweating.
  • thrombocytopenia, masauki disturbances, erythema multiforme, mydriasis, Stevens - Johnson, na gani disturbances, illa dandano, da tsawaita na zub da jini lokaci, wani rauni, fata na gaggawa, gajiya, anaphylactic halayen.

Ya kamata kuma a lura da cewa, bayan da na ba zato karbo daga cikin la'akari abin hawa ko rage sashi ne yiwu wannan gefe halayen kamar yadda juyayi irritability, gajiya, zawo, drowsiness, restlessness, ciwon kai, paraesthesias, tashin zuciya, hypomania, amai, sweating, anorexia, rashin barci, bushe bakinka, juyayi, dizziness da kuma disorientation. Yawanci, wadannan cututtuka su ne m kuma tafi ba tare da wani magani.

shawarwari

Sayar ko antidepressants ba tare da takardar sayen magani? A jerin wadannan magunguna ba sosai babban ( "Prozac", "Paxil", "Despres", "Azafen", "Persian", "amitriptyline"), da kuma miyagun ƙwayoyi "Velaksin" ba kunshe a shi. Saya shi a Pharmacy, za ka iya kawai ta ganin likita.

Kafin shan wannan magani karkashin review, musamman marasa lafiya da depressive cuta, ya kamata a yi la'akari da wani babban yiwuwa na kunar yunkurin. A wannan batun, a farkon miyagun ƙwayoyi far shawarar don amfani a cikin m kashi da kuma karkashin kusa likita dubawa.

Mutane da yanayi cuta a lokacin jiyya da antidepressants iya ci gaba manic ko hypomanic jihar.

Marasa lafiya ya tabbata dõmin ya yi gargaɗi da bukatar nan da nan ganin likita idan akwai urticaria abubuwa, rashes ko rashin lafiyan halayen.

Wasu marasa lafiya a kan aiwatar da samun venlafaxine kiyaye kashi-dogara karuwa a jini.

Tsofaffi da marasa lafiya ya kamata a yi gargadin da wani yiwu take hakkin da hankali na auna da kuma dizziness ci gaba.

A lokacin jiyya da na kudi kamata kauce wa shan giya.

Antidepressant "Velaksin": haƙuri shedu, samfurin analogues

Abin da mutane suke cewa game da wannan miyagun ƙwayoyi zuwa wani haƙuri? Mutane da yawa masu amfani da sun ruwaito wani babban yawan illa cewa faruwa yayin da shan wannan magani. Sau da yawa sosai da wannan magani Yanã m halayen kamar drowsiness, wani rauni, rashin barci, seizures, mahaukaci tunani, ciki da kuma rikice. Bugu da kari, wasu marasa lafiya da'awar cewa wadannan effects kasance bayan kammala magani. Har ila yau, da yawa masu amfani koka game da bayyanar janyewar bayyanar cututtuka da kuma dogaro.

Abin da zai iya maye gurbin antidepressant kamar "Velaksin"? Analogs wannan magani ba za a samu a duk drugstores. Matsayin mai mulkin, masana Wadannan sun hada da wadannan: "Venlafaxine Sandoz", "Efevelon", "Alvent", "Nyuvelong", "Velafaks", "Dapfiks", "Voksemel", "Venlaksor", "Vensuert", "venlafaxine".

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