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Da miyagun ƙwayoyi "Captopril" daga abin da? Aikace-aikace, reviews, farashin

Abin da ake da miyagun ƙwayoyi "Captopril", daga abin da aka yi amfani da da kuma abin da kaddarorin? A amsa ga dukkan wadannan tambayoyi za a iya samu a cikin kayan da wannan labarin. Bugu da kari, za mu gaya muku game da yadda za a dauki da miyagun ƙwayoyi da kuma abin da illa, kuma contraindications ga yin amfani da shi yana da.

Janar bayani game da magani samfurin

Drug "Captopril" a Latin sauti kamar "Captopril". Wannan magani ne a roba hanawa na angiotensin-tana mayar enzyme (ACE ko rage tsawon). Ya yi amfani da ko'ina a cikin likita yi, to hanzari rage jini.

A abun da ke ciki da kuma tsari da miyagun ƙwayoyi saki

Medicament "captopril" - daga wanda da kayan aiki da ake sa wa? Yawanci, likitoci rubũta ta ga waɗanda suke kullum fama da hauhawar jini. Gabatar ana sayar da maganin kawai a cikin wani nau'i na spigot Allunan cewa an sanya shi a cikin kartani. The aiki sashi na wannan miyagun ƙwayoyi ne captopril. Da abun ciki a cikin kowane kwamfutar hannu ne 25 ko 50 MG. Daya kunshin iya zama 100, 50, 40, 30, 20 ko 10 na fadiwa.

A pharmacological mataki da miyagun ƙwayoyi

Kamar yadda aka tattauna a sama, "Captopril" Allunan umurci wanda aka nested a kartani, shi ne wani mai hanawa na angiotensin-tana mayar enzyme (ACE Ina nufin).

Ya kamata a lura cewa antihypertensive kaddarorin da miyagun ƙwayoyi suna hade da m hanawa na ACE aiki, abu don wani gagarumin raguwa kudi hira angiotensin 1 ga angiotensin 2, wanda shi ne wani fairly m vasoconstrictive bangaren.

Bayan wani gagarumin raguwa a cikin taro na angiotensin 2 ne a maimaita karuwa a jini renin aiki ta kawar da mummunan feedback idan aka saki, da kuma kai tsaye akan rage aldosterone samar. Bugu da kari, da medicament "Captopril", analogs wanda aka gabatar a nan, na iya tasiri da kallikrein-kinin tsarin, game da shi, da hana rugujewar bradykinin.

Saboda da vasodilating sakamako daga cikin miyagun ƙwayoyi muhimmanci rage jimlar jijiyoyin bugun gini juriya (gefe), capillary sandan matsa lamba da kuma huhu jijiyoyin bugun gini juriya a gare su. Bugu da kari, shi ne iya ƙara da minti girma daga cikin zuciya tsoka da kuma motsa jiki haƙuri.

Idan da miyagun ƙwayoyi "Captopril", reviews daga waxanda suke da mafi kyau, kai mai dogon lokaci, shi ya hana a ci gaba da zuciya rashin cin nasara, rage tsananin tsokar hypertrophy na hagu ventricle, kazalika da jinkirin saukar da ci gaban dilation.

Bugu da kari, da medicament ne iya hana ci gaban m nephropathy, ragewan sautin efferent koda arterioles, kuma glomeruli muhimmanci inganta intraglomerular hemodynamics.

Pharmacokinetics da miyagun ƙwayoyi

Bayan shan miyagun ƙwayoyi a ciki ya sauri tunawa. Aiki da wani medicament fara bayan game 40-60 minti. Matsakaicin taro an samu a cikin jikin mutum bayan na farko da awa daya.

Ya kamata a lura da cewa lokaci daya ci abinci tare da ba magani na rage absorbability na 30-40%. Wannan shi ne dalilin da ya sa Allunan rika dauka a kan 1 hour kafin cin abinci ko bayan 1-1.5 hours bayan haka.

Duration na mataki bayan yin amfani da medicament (domin su runtse jini) ya dogara da multiplicity na ta liyafar da kuma sashi. Ga ci gaban da cikakken warkewa sakamako mai haƙuri iya bukatar makonni da dama na far.

Halaye da kuma kaddarorin da miyagun ƙwayoyi "Captopril"

Yanzu ka san cewa shi ne mai magani "Captopril", daga abin da aka yi amfani da da kuma yadda za a yi aiki dangane da jikin mutum. Amma don gane dalilin da yasa wannan magani ne don haka rare, ya kamata ka yi la'akari da kaddarorin.

The aiki abu wanda yake shi ne wani ɓangare na "Captopril" shiri mallaka vasodilating, antihypertensive da cardioprotective Properties.

Wannan magani ne iya kara saki na ilimin aiki abubuwa da cewa suna da wani natriuretic sakamako. Saboda wannan dukiya muhimmanci inganta jini ya kwarara zuwa kodan. Bugu da kari, da medicament "Captopril" na matsa lamba da kuma rage total post-preload a zuciya, da kuma ƙaruwa a cardiac fitarwa.

Alamomi ga yin amfani da miyagun ƙwayoyi

Gabatar magani nuna domin lura da wadannan munanan:

  • Jijiya hauhawar jini da kuma renovascular. Yana za a iya amfani da a hade ko a matsayin monotherapy.
  • Cuta na hagu ventricle. Yawanci, da miyagun ƙwayoyi da ake amfani da mutanen da suka yi a zuciya da kuma yanzu a asibiti barga yanayin.
  • M nephropathy. Sanya kawai ga waɗanda suka yana da ciwon sukari farko type, watau insulin-dogara mutane.
  • Cardiomyopathy.

Drug "captopril" - daga abin da kuma ake sa wannan magani? Kamar yadda aka sani, da miyagun ƙwayoyi za a iya gabatar da amfani a cikin hadaddun far da zuciya rashin cin nasara (congestive).

Contraindications don yin amfani da medicament

Bisa ga umarnin, da miyagun ƙwayoyi "Captopril" da aka tsananin haramta wa kai a cikin wadannan lokuta:

  • A hali na hypersensitivity zuwa aiki sashi - captopril. Ya kamata kuma a lura da cewa aiki miyagun ƙwayoyi ba da shawarar ga wadanda suka yi wani rashin ha} uri, akwai wani sarari kungiyar da kwayoyi, wanda suke hanawa na angiotensin-tana mayar enzyme (Ina nufin, marasa lafiya da suke raya angionefrotichesky kumburi a lokacin jiyya da sauran ACE hanawa).
  • Lokacin da ya bayyana adam hanta aiki.
  • A cardiogenic buga.
  • Lokacin da narkewa kamar fili cuta.
  • Lokacin da ya bayyana adam koda aikin yanayin bayan dasawa na gaba, tsakanin stenosis na jijiya, azotemia, hyperkalemia, kuma primary hyperaldosteronism.
  • Idan hypotension.
  • A immunological cututtuka.
  • Mitral stenosis da aortic stenosis.

Bugu da kari, da miyagun ƙwayoyi "Captopril" analogues na wannan magani ba da shawarar ga mata masu ciki, yara a karkashin shekaru 18 da haihuwa, kazalika da masu jego.

Drug "Captopril": wa'azi, farashin magani

Bisa ga a haɗe umarnin, da miyagun ƙwayoyi ya kamata a dauka game da 1 hour kafin abinci. A tsawon lokaci da far da kuma sashi regimen magani gabatar ya kamata a ayyana kawai likita a kan wani mutum-akai, dangane da irin da ya kwarara daga data kasance cuta.

Saboda haka yadda za a yi da miyagun ƙwayoyi "Captopril"? Kashi (na farko) na medicament a cikin ganewar asali da hauhawar jini ne 12.5 MG sau biyu a rana. A m bukatar lokaci daya za a iya amfani da shiri na 2 Allunan na 25 MG. Amma a wannan yanayin da liyafar ne kyawawa da za a rarraba su zuwa sau 3. A kalla kullum kashi na irin wannan medicament ne 150 MG.

Idan likitan ka ya ya wajabta tabbatarwa far na dogon lokaci, da magani "Captopril", wanda shaidan mu sake nazari kawai sama, ya yi ta farko kwamfutar hannu (25 MG) sau uku ko sau biyu a rana.

Lokacin da renovascular hauhawar jini da kuma na koda farko sashi na medicament ne 6,25 MG sau uku a rana. Taimaka far kamata hada da wani 1 kwamfutar hannu halitta (25 MG) sau uku a rana.

Idan kana kamu da kullum zuciya da kuma gazawar akwai magudi a kodan, da farko sashi ya zama 12.5 ko 6,25 MG sau uku a rana. Kamar haka kowane 2-3 makonni ya kamata a kawo ta tabbatarwa kashi na 25-50 MG, tare da wannan mita. Mai karɓa Hanyar postinfarction tsawon medicament kama.

ACE kungiyar da kwayoyi a cikin tsofaffi an sanya kawai ga ilimin. A wannan yanayin, da magani ya kamata a individualized. Karɓi "Captopril" wadannan mutane ya kamata ya zama m kashi. Bugu da kari, an ba da shawarar kara a ko'ina cikin magani. Lokacin da cikakken zama dole, za ka iya bugu da žari amfani da madauki diuretic.

Amma ga farashin, sa'an nan for 40 Allunan na wannan samfurin ka zai biya game 50-60 Rasha rubles. Kamar yadda ka gani, yana nufin "Captopril" ne mai gwada m miyagun ƙwayoyi da yadda ya kamata ƙananan jini a da lafiya hanya.

Dauka tare da matsananci hankali

Gabatar magani ya kamata a dauka tare da matsananci hankali a lokacin da:

  • hanawa na bargo jini wurare dabam dabam.
  • m autoimmune cututtuka.
  • ciwon sukari.
  • cerebral ischemia .
  • jijiyoyin zuciya da cututtukan zuciya.

illa

Bisa ga umarnin, bayan da miyagun ƙwayoyi "Captopril" na iya faruwa a marasa lafiya wadannan gefen halayen:

  • bronchospasm, mashako, shortness na numfashi, bushe unproductive tari.
  • CNS ciki, da ciwon kai, seizures, ataxia, juwa ko jiri, tingling a cikin manya da ƙananan extremities, kazalika da ji na numbness, da ruɗewa, disturbances na wari da kuma hangen nesa, gajiya, ciki;
  • exfoliative dermatitis, itching, fata na gaggawa, photodermatitis, pemphigus, angioedema, urticaria, anaphylactic buga, mai guba epidermal necrolysis, alopecia.
  • zuciya kari disturbances, angina pectoris, orthostatic hypotension, tsokar zuciya infarction, tachycardia.
  • dandano tashin hankali, flatulence, asarar ci, stomatitis, tashin zuciya, maƙarƙashiya, glossitis, ulcerative raunuka na ciki mucosa da bakinka, zawo da amai, xerostomia, ciwon mara.
  • paresthesia, amosanin gabbai, na gefe neuropathy.
  • neutropenia, hyperkalemia, thrombocytopenia, agranulocytosis, eosinophilia.
  • oliguria, proteinuria, sosai koda aiki.
  • cholestatic hepatitis, pancreatitis, cholestasis, hepatocellular necrosis.

A cewar martani da cewa bar masu amfani da wannan magani, illa iya faruwa yafi idan, yayin da shan magani don cika da low-gishiri ko gishiri-free rage cin abinci.

Drug "Captopril": yawan abin sama

A yawan abin sama data nufin marasa lafiya na iya bayyana illa kamar tsokar zuciya infarction, da kuma bayyana ta a m drop a jini, m tashin hankali na cerebral wurare dabam dabam da kuma thromboembolic rikitarwa.

rigakafi

A cewar masana, shi ba da shawarar a yi da miyagun ƙwayoyi da potassium-sunã rãyar da diuretics, da sauran kwayoyi da muhimmanci ƙara da taro na potassium a cikin jini jini. Idan muka yi watsi da wannan Council, akwai babban hadarin hyperkalemia.

Bugu da kari, da miyagun ƙwayoyi "Captopril" ya kamata a yi amfani da tare da matsananci hankali tare da lokaci daya liyafar nufin "Procainamide", "" allopurinol "," Azathioprine "ko wasu immunosuppressants, musamman a cuta da na koda aiki.

A yaxuwa connective nama cututtuka, kazalika da kullum zuciya rashin cin nasara, da miyagun ƙwayoyi da bukata kawai da za a dauka a karkashin kusa likita dubawa.

Ya kamata kuma a lura da cewa, bisa ga likita da marasa lafiya da kuma sake dubawa, da hypotensive sakamako na medicament rage miyagun ƙwayoyi "Indomethacin" da kuma estrogens.

ajiya yanayi

Drug "Captopril" yana nufin kwayoyi List B. Wannan magani an saki a kantin sarƙoƙi kawai a kan ganin likita. Its shiryayye rayuwa ne shekaru 3 daga ranar yi. Irin wannan hanyar dauki zai fi dacewa a cikin duhu da kuma bushe wuri, a zazzabi ba wucewa 25 ° C.

miyagun ƙwayoyi analogues

Bisa ga aiki sashi yana da wadannan tsarin analogs wannan magani:

  • "Captopril Verein".
  • "Angiopril-25".
  • "Captopril Acre".
  • "Alkadiene".
  • "Captopril Sandoz".
  • "Vero Captopril".
  • "Captopril UBF".
  • "Blokordil".
  • "Captopril Akos".
  • "Captopril hexane".
  • "Capoten".
  • "Captopril FPO".
  • "Captopril Sar".
  • "Katopil".
  • "Aegis Captopril".
  • "Epsitron".
  • "Captopril STI."

Kamar yadda ka gani, ƙaddamar magani yana da quite 'yan musamman. Saboda haka, sau da yawa marasa lafiya kiwata tambaya ga abin da yake mafi alhẽri - da miyagun ƙwayoyi "Captopril" ko "Capoten". A babba bambanci tsakanin su. Sun bambanta daga juna kawai da manufacturer. A saboda wannan dalili, yana nufin "Capoten" da daraja 3.5 sau mafi tsada miyagun ƙwayoyi "Captopril".

Sharhi kan shirye-shiryen

Duk da low price, da medicament "Captopril" yadda ya kamata lowers jini. Marasa lafiya da suke yi akai-akai amfani da wannan magani ce cewa ta effects bayyananna a cikin 1-3 hours bayan ingestion.

Mutum rashin lafiyan halayen bayan aikace-aikace na wakili faruwa a game da 5-8% na mutanen da. Mutane da yawa jayayya da cewa wannan magani sa mai tsanani kumburi. Wannan shi ne dalilin da ya sa kafin amfani, a tabbatar shawarci tare da likita. Idan da wajen "Captopril" shi ne akalla daya gefen sakamako, yana da kyawawa don ki daga shi kuma tafi a kan wata warkewa ga hawan jini daga wata ƙungiyar.

Akwai quite mai yawa reviews cewa "Captopril" kwayoyi "Capoten" da sauran analogues na wadannan kudi yadda ya kamata taimaka wajen rabu da hauhawar jini tsofaffi. Amma kafin wannan wata dabara, a tabbatar shawarci tare da likita. Bugu da kari, da mutum a cikin tsufa don kawar da cutar hawan jini da kuma sauran cututtuka bada shawarar yin amfani kawai da mafi ƙasƙanci kashi na magani.

Shin shi mai lafiya don amfani da miyagun ƙwayoyi?

Bisa ga yankin asibiti a Rivne (Ukraine) a 2010, da wani binciken da aka gudanar mita na illa daga shan miyagun ƙwayoyi "Captopril". A wannan hanya, ya samu halartar mutane da m kuma matsakaici jijiya hauhawar jini. A sakamakon haka, na 500 batutuwa koka da illa kawai mutane 73. Daga cikin wadannan, 53 - daina shan miyagun ƙwayoyi, da kuma sauran 20 - ci gaba, kamar yadda suka gano cewa, shi ya kawo mai yawa fiye da kyau fiye da cutar da lafiya.

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