Kiwon lafiyaShirye-shirye

"Montelukast": reviews, umarnin da analogues da miyagun ƙwayoyi

"Montelukast" - game da miyagun ƙwayoyi da sake dubawa za a iya samu a online forums da kuma shafukan kwazo da matsalar fuka - wani classic antagonist na leukotriene D4-tsoka mai amsa sigina. Da miyagun ƙwayoyi ne yadu amfani matsayin tushe a lokacin far da su hana halayyar hare-haren da cutar. Daidaita abun da ke ciki da damar yin amfani da wani magani domin lura da marasa lafiya na kusan kowane zamani kungiyar.

saki Form

Dalilan da ya sa "montelukast" samu mafi yawa m reviews, mai yawa. Duk da haka, abu na farko da cewa kama da ido - wannan shi ne, ba shakka, wani tsari na Allunan, sayar karkashin cinikin sunan data.

A lokacin da tsari aka mamaye uku matrix. Shi ne game da misali kwayoyi tare da tsare ambulan (1 naúrar ƙunshi 10 MG na aiki abu) da kuma su analogues taban da ake (4 MG da 5 MG daidai da na reagent). Base akai a lokuta biyu, abubuwa montelukast sodium, amma abun da ke ciki na dama daban-daban karin aka gyara - mannitol da aspartame ne ba a samfurori nufi ga nan da nan ingestion a lokacin amfani.

A comments quite sau da yawa shi baba up tambaya na counterfeits, wanda a yanzu da kuma nan ya bayyana a kantin sarƙoƙi. Kare da kayayyakin na jabu iya zama, idan ba dace kula da bayyanar da pharmacological samfurin.

A musamman, taban da ake kwaya da 4 milligrams na aiki sashi, yana da wani m siffar da kuma mai ruwan hoda tinge (bayanin yayi dace Allunan da ceri dandano, tare da yin amfani da wasu flavorings halatta bambance-bambance), da kuma alama da lambobin "4" a gefe daya. Analogs a cikin abin da babban aiki sashi ne 1 MG more - zagaye da suna "biyar". Kwayoyi a matsayin harsashi geometrically kama wani murabba'i mai dari. Su m da ya ƙidaya "10" lambar.

pharmacological akidar

"Montelukast" (nassoshi kwatanta yanayi inda hadaddun reagent tsokani allergies ne musamman rare) - wannan shi ne wani hali wakilin kungiyar antibronhokonstriktornyh kwayoyi. A algorithm damar ayyukansa yi magana da wani "dangantaka ta kusa" tare da intermedianty / prostaglandins da thromboxanes.

Babban aiki na da miyagun ƙwayoyi - tarewa cysteinyl leukotriene "na'urori masu auna sigina" na numfashi tsarin. Wadannan rabe tsare high aiki a Bronchial fuka ci gaba da kuma su ma ta da kira na secretions wanda sa'an nan accumulates da kuma dagula mucosa.

Regular ci kaiwa zuwa wani gagarumin raguwa a cikin tsanani daga cututtuka a bango na janar karu a yawan fuka-haren (kamar yadda muka gani da yawa marasa lafiya, m canje-canje riga lura a farkon zamanin far).

rayuwa siffofin

"Montelukast" (reviews harhada magunguna bayar da shawarar cewa real zabi na tsayawar-ins yana da iyaka ga farashin siyasa na masana'antun, watau mutum kwayoyi-ma'ana, yana nufin abun da ke ciki m-tsari kwayoyin ne babban bangaren, akwai sau da yawa ya fi tsada fiye da bayyana shirye-shiryen), shiga jini jini, ta ɗaure da daidai da ta sunadarai. A asibiti karatu, sakamakon da aka rubuta a 99, 37%. A lokaci guda, ta bioavailability ne a kai tsaye gwargwado ga aiwatar da bayar. Alal misali, da sinadaran 5-milligram Allunan amenable zuwa sha da 73%, alhãli kuwa analogues da membrane shafi a cikinsa akwai sau 2 more aiki abubuwa, - kawai da 64%.

A irin wannan halin da ake ciki tare da rabin-rai na reagent: Aka gyara taban da ake kwayoyi, ta jurewa metabolism, da barin jiki bayan 2 hours bayan liyafar, amma bijiro da batun kafa abubuwa na al'ada Allunan - bayan 180-200 minti. A wannan jini yarda dabam tsakanin 43-45 ml / minti daya. Kuma, sha'awa, kawai 0.2% na kashi ne ya isar urinary tashoshi. Hanji, ta kwatanta, - fiye da 85%.

Daga cikin comments na girmamawa hukuma, shi ya bi da cewa pharmacokinetic tsari ne daidai da smoothly a marasa lafiya na biyu mata da maza, da cewa yin wasu tsanani sabawa for shekaru da kuma na koda Pathology a cikin lissafi na kullum servings magani ake bukata. Amma da gazawar da hanta, musamman a lokacin da ta je ga mai tsanani cuta, ya cancanci kulawa ta musamman a cikin shirye-shiryen da wani warkewa jadawalin.

alamomi ga

Lokacin da barata ta wurin yin amfani da "montelukast" miyagun ƙwayoyi reviews (yara magani shawarar a cikin nau'i na danko, kwayoyi, mai rufi membrane harsashi, shi ne bu mai kyau ya nada kawai manya da matasa), bar a kan Forums, ba shakka, taimake mu mu fahimci. Duk da haka, kawai shiryar da sauran mutane ta ra'ayi - shi ne babban kuskure, saboda ba tare da shawara tare da likita, "a gane" irin fuka, da kuma mafi muhimmanci - don gano dalilan da ya faru shi ne kusan ba zai yiwu.

Game da hukuma sanarwa, cikin da'irar akwai cututtuka, ailments da sauran yanayi kayyade kamar haka:

  • Bronchial spasms jawo ta wuce kima jiki kaya;
  • Yanayi / kullum rhinitis, rashin lafiyan yanayi na asalin;
  • asma.
  • da bukatar m matakan.

A ganiya sashi

"Montelukast" (korau feedback ne musamman wuya a sami, saboda aiki sashi ya dade da aka samu nasarar yi amfani da matsayin core bangaren da yawa miyagun ƙwayoyi) da aka gudanar da baki, sau daya a rana, ba tare da yin wani jadawalin "karin kumallo - abincin rana - abincin dare."

Domin chewable Allunan, 4 MG da 5 MG ne irin dosages sharudda:

  • yara shekaru tsakanin 2 da 5 shekaru: 1 naúrar samfur (4 MG) a rana, a lokacin kwanta barci, har cimma iko da cututtuka da kuma tsawaita na wajibi Hakika for 2-4 makonni a gyara resultant sakamako.
  • marasa lafiya 6 zuwa shekaru 14 da haihuwa: wannan yanayin, amma a daya-lokaci kudi na - 5 MG.

Domin kwayoyi tare da tsare wrapper dacewa wadannan shawarwari:

  • manya da yara a kan shekaru 15 da haihuwa, na fama da Bronchial fuka ko na kullum rhinitis: 1 Unit (10 MG na abu) / rana da yamma.
  • su hana cramps: wannan kashi a kan wani lokaci tazara tsawon 14-28 kwanaki.

gefen sakamako

"Montelukast" wa'azi (reviews bayar da shawarar cewa ko da a full yarda da hukuma jagorancin atypical halayen ga gaban sinadaran zuwa karshen ba za a iya cire) tana wurinta a matsayin yiwuwar hadari miyagun ƙwayoyi, amma tare da proviso cewa ba takamaiman "mayar da martani" a kan sashi na jiki a cikin mutum lokuta har yanzu zai yiwu.

Halatta labari:

  • GI: zawo, bushe baki, zafi a ciki ciwo, tashin zuciya.
  • zuciya da kuma jini Lines: wani sosai gagarumin karuwa a bugun jini kudi.
  • fata rash, urticaria, gida hematoma.
  • numfashi tsarin: runny hanci da tari.
  • CNS: dizziness, gajiya, yanayi na ciki alternating da matsanancin psychomotor agitation.
  • musculoskeletal: myalgia da arthralgia (ciki har da convulsions.).
  • Sauran: cututtuka halayyar m na numfashi cututtuka da kuma mura.

Gazawarsu da kuma contraindications

"Montelukast" (umarnin don yin amfani da shi ne mafi kyau sake dubawa, da kuma bayanai na dauke da shi, a cikin sharuddan objectivity, tambayoyi daga 'yan forum ne kusan ba akwai) za su shafi idan:

  • Yana samu wani ƙara ji na ƙwarai to abun da ke ciki na magunguna (kullum na gaskiya ga duk iri Allunan).
  • bincikar lafiya rare gaji cuta, ciki har da waɗanda suke a wanda kwayoyin ba assimilate galactose ko fuskantar mawuyacin lactase rashi (wannan hanin bai shafi taban da ake kwayoyi).
  • da haƙuri da aka nauyaya phenylketonuria.
  • da mãsu haƙuri ya ba tukuna juya shekaru biyu (ga mai rufi Allunan "shekaru iyaka" - 15 years).

Yawan abin sama: Bayyanar cututtuka da kuma Jiyya

Nazarin ya nuna, "Montelukast" 4 MG (nassoshi game da wannan ciniki irin na reagent, a gaskiya, m ga comments cewa suna magana ne taban da ake analogs dauke 5 MG na aiki abu) a wuce haddi na da kullum amfani rate yana a kan wannan sakamako kamar 10 MG Allunan . A mafi furta bayyanar cututtuka na yawan abin sama za a iya gani a marasa lafiya ƙaramin rukuni. Manya, ko da shan 200 MG / rana domin 5 months, wasu mahaukaci halayen da aka kiyaye.

The guda alamar aukuwa na ƙãra yawa da miyagun ƙwayoyi ne:

  • unquenchable ƙishirwa.
  • drowsiness.
  • ciki yankin zafi.
  • amai.

Jiyya ne da za'ayi, dangane da asibiti hoto kiyaye. Bayani game da tasiri na hemodialysis fakowa ba.

Drug interactions, kuma mafi mashahuri analogues

"Montelukast" 5 MG (reviews na taban da ake samfurori bar ta pediatricians, tafasa saukar da ra'ayin cewa da miyagun ƙwayoyi, babu shakka, ya cancanci hankalin matasa iyaye), kazalika da sauran siffofin leukotriene tsoka mai amsa sigina antagonist, a lokacin da amfani da, a layi daya da dacewa jamiái su hanzarta da kyau kuzarin kawo cikas : cututtuka na fuka zama kasa mai tsanani, da yawan hare-hare rage. Duk da haka, da ba zato karbo daga far da za'ayi a kan tushen da inhaled corticosteroids ba da shawarar.

Muhimmanci saɓani a cikin pharmacokinetic matakai shafe theophylline da prednizola gano. Amma sha a "ƙungiyar" tare da phenobarbital raguwa da kamar yadda 40%.

Reagents cewa hana kira na CYP3A4 isoenzyme, ya kamata a yi amfani ne kawai a karkashin likita dubawa.

Tsarin analogs cewa an fi sau da yawa samu a sale:

  • "Monkasta".
  • "Singlon".
  • "Singulair".
  • "Ektalust".
  • "Singuleks".

"Singulair" ko "montelukast": reviews na likitoci da kuma harhada magunguna

Kamar yadda gwani pharmacologists, muhawara game da abin da na kwayoyi ne mafi aminci kuma mafi inganci, ma'ana, tun "Singulair" da "montelukast" ne daya da kuma guda pharmaceutical tushe. Just wuce na farko cinikayya sunan patent rajista, da kuma na biyu shi ne na kasa da kasa. Mutane daya-daya da kuma likitoci da marasa lafiya, duk da haka, daukan wani daban-daban view kuma la'akari da magani aka rarraba ƙarƙashin INN, kadai daidai yanke shawara.

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