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Da miyagun ƙwayoyi "Novocaine": umarnin don amfani, farashin. "Novocaine" a ciki

Medicine "Novocaine" shi ne wani tasiri analgesic miyagun ƙwayoyi. Magani a kan jerin mafi muhimmanci na'urorin kiwon lafiya.

Pharmacological Properties "Novocaine" miyagun ƙwayoyi

Umurnai na amfani na nuni da cewa da miyagun ƙwayoyi yana da wani gida m matsakaici aiki, an yi amfani da ko'ina a cikin likita yi. Shiri "Novocaine", wanda yake shi ne mai rauni tushe, sodium tashoshi suna katange da inhibiting da ci gaba da kuma yada jijiyar a jijiya zaruruwa da endings. Lokacin karbar medicament effects wani canji na iko a neuronal Kwayoyin, tare da gagarumin rinjayen a kan Allaha m ba a bayar. Da miyagun ƙwayoyi cike yaduwa daga zafi hasken dake fitowa.

A lokacin da tsotsa kuma nan da nan ta shiga cikin jini a lokacin da gudanar intravenously akwai wani karu daga excitability na gefe cholinergic tsarin, da kuma rage haifuwa na a saki acetylcholine preganglionic endings. A medicament "Novocaine" (umurci manual bayani game da wannan) gusar spasms of m tsoka, rage excitability na mota yanki na kwakwalwa bawo da infarction.

Domin igiyar jini amfani, da mafita yana da antiarrhythmic, hypotensive, antishock, analgesic sakamako, qara tsaurin lokaci, muhimmanci rage da watsin, kuma automaticity excitability. A amfani da high allurai na iya faruwa a take hakkin da juyayi tsoka madugu, convulsions an kiyaye.

A magani kawar da birki da downward tasiri na kwakwalwa kara, wani depressing sakamako a kan polisinapticheskie reflexes. Yana yana da wani gajeren m aiki. Action infiltration maganin sa barci yana daga minti 30 zuwa awa 1. The bayani "Novocain" gabatar intramuscularly tsofaffi da marasa lafiya a farkon matakai na pathologies iya yadda ya kamata yaki da cutar hade tare da mai illa aiki na juyayi tsarin, cerebral spasms, jijiyoyin zuciya da kuma jijiyoyin bugun gini hauhawar jini.

Da miyagun ƙwayoyi ne talauci tunawa a cikin mucous. Lokacin da aiki wakili sauri allura a cikin jini, an hydrolyzed da esterases tsokoki da kuma jini, forming biyu babban aiki metabolite: PABA (antagonists da tsoka shan kwayoyin sulfa) da kuma diethylaminoethanol (da ciwon matsakaici vasodilating mataki). Nuna a kodan a cikin nau'i na metabolites.

A abun da ke ciki da kuma nau'i na "Novocaine" miyagun ƙwayoyi

Samar da miyagun ƙwayoyi a matsayin mafita ga allura ne bayyananne, colorless ruwa, a ampoules girma daga 1 zuwa 20ml. A kashi na aiki sashi a cikinta shi ne 0.25 da kuma 0.5. Bugu da kari, daya- da biyu-kashi saki "Novocaine" shiri bayani. Farashin wannan tsari ne game da 15 rubles.

Popular kuma foda, kazalika da bakararre bayani daga medicament, zuba a cikin vials na 0.2 da kuma 0.4 lita. Domin lura da yawa cututtuka tambaya shafawa 5 da kuma kashi 10, da kuma suppositories, wanda dauke da 0.1 grams na aiki sashi (procaine hydrochloride), kazalika da karin aka gyara - witepsol ko tallow. A 1 ml na wani aiki abu dauke a cikin adadin 0,005 grams, ƙarin aka gyara aiki hydrochloric acid da kuma ruwa ga allura.

alamomi

Drug "Novocaine" umarnin don amfani da ake karfafa su gabatar da yin retrobulbar, m, laka, waya, epidural, infiltration maganin sa barci. Amfani medicament kayan vagosympathetic da perirenal lakar kawancen. Aikace-aikace na suppository ne tasiri ga analgesia da tsuliya fissures da haemorrhoids. Amfani da man ƙanshi ya sa bayyanar cututtuka na neurodermatitis, eczema, itching dermatosis.

Medicine "Novocaine": umarnin don amfani da

Injections adult marasa lafiya kamar yadda ka yi infiltration maganin sa barci a wani juz'i na 300-600 MG (0.25-0.5 kashi bayani).

M da rarrafe infiltration Wisniewski hanya ake yi ta hanyar gabatar 0.25% bayani a cikin wani adadin 125 ml. Epidural maganin sa barci da aka yi tare da taimakon "Novocaine" biyu-kashi bayani. Injections jagora ya bada shawarar a sashi na 25 ml. Kashin baya maganin sa barci samu ta hanyar 2-3 ml na 5% miyagun ƙwayoyi. A ENT yi 10% daga cikin miyagun ƙwayoyi bayani da ake amfani da Topical maganin sa barci.

Don kara tsawon lokaci na mataki na miyagun ƙwayoyi da kuma rage absorbability, kuma ma a wani gida m miyagun ƙwayoyi "Novocaine" diluted bayani daga epinephrine hydrochloride. Don yi da electrophoresis bada shawarar yin amfani da wani 10% miyagun ƙwayoyi. A perirenal kitse a lokacin da kawancen na Wisniewski dole ka shigar da 60 ko 120 ml na 0.5-th ko 0.25% bayani, bi da bi. Vagosympathetic kawancen samar da gabatar da 100 ml na samfurin na 0.25% taro.

Duk da contraindications injections "Novocaine" yara sukan wajabta a matsayin analgesic a lokacin da gwamnati da sauran magunguna. A sashi da aka lasafta bisa ga nauyin da yaro (ba fiye da 15 milligrams da kilogram).

Rectal suppositories ana amfani da bayan a baya ya yi purgation via enema ko ta halitta. Lokacin da fata pathologies Maganin shafawa amfani da shafa bakin ciki Layer rufe biyu sau a karan.

illa

Drug "Novocaine" (umarnin don amfani gargaɗi da wannan) na iya haifar da mummunan halayen.

Tsakiya da kuma na gefe m tsarin amsa da magani ciwon kai, wani rauni, drowsiness, juwa ko jiri, restlessness, seizures. A wasu lokuta, akwai wani tremor, asarar sani, lockjaw, ji kuma na gani hanawa, paraesthesia, inna da kafafu, nystagmus. Bugu da kari, akwai iya zama numfashi inna, tarewa da numfashi tsokoki.

Cardio-jijiyoyin bugun gini tsarin ne wani canji a jini, akwai zafi a cikin kirji, arrhythmia, bradycardia, auka, na gefe vasodilatation.

Urinary da kuma narkewa kamar tsarin amsa magani amfani involuntary urination, defecation, amai da kuma tashin zuciya.

A wani ɓangare na jijiyoyi da illa hada methemoglobinemia. Bugu da kari, da miyagun ƙwayoyi zai iya sa rashin lafiyan halayen:

  • amya.
  • anaphylaxis .
  • fata rash.
  • itching.

Ga wasu korau halayen hada da m maganin sa barci, rashin ƙarfi, hypothermia, ciwon baya. A lokacin maganin sa barci a Dentistry lura tsawon kwanakinka da maganin sa barci, paresthesia da numbness na lebe da kuma harshe.

yawan abin sama

Don amfani da "Novocaine" miyagun ƙwayoyi sayen magani, wanda ya nuna da magani regimen ya kamata a wajabta ta likita. Gaza bada hašin kai dokokin iya zama alamun wani yawan abin sama. Bayyanar cututtuka na wuce kima amfani da medicament ne pallor na mucous membranes da kuma fata integument, methemoglobinemia, apnea, kwatsam matsa lamba maniyyi, tachycardia, shortness na numfashi, amai, sanyi rika zufa, tashin zuciya, juwa ko jiri. Marasa lafiya da hankali na tsoro, motor agitation, convulsions, hallucinations. Domin kawar da manifestations na yawan abin sama, dole a gudanar da wani na huhu iska tare da oxygen inhalation, a halaye da wuya, rubũta symptomatic da detoxification far.

contraindications

Amfani da miyagun ƙwayoyi yiwu ba dukan marasa lafiya. Lokacin da maganin sa barci hanya haramta masu rarrafe infiltration wakili don nama fibrotic canje-canje. Subarachnoid maganin sa barci ba za a iya da za'ayi a wata septicemia, bugu jihohi, hypotension, zub da jini. An ba da shawarar tafiyar da na yau da kullum da magani, misali, yin damfara da "Novocaine".

Tare da hankali shiri amfani a lokacin da gudanar da marasa lafiya da m jini hasara, koda gazawar. ga yanayin shafe akan rage hanta jini wadata, m cardiac da jijiyoyin bugun gini insufficiency. a kan kamuwa da cuta a cikin allura site. kumburi pathologies. Karkashin musamman likita dubawa wajibi ne a yi amfani da magani a lokacin haihuwa, nauyi da kuma debilitated marasa lafiya, tsofaffi mutane da kuma yara yan kasa da shekaru rinjaye.

Tare da hada magani tare da anticoagulants ( "danaparoid" "Warfarin", "Ardeparin", "dalteparin", "Enoxaparin" "Heparin") na kara hadarin zub da jini. Ragewan da matsa lamba da kuma bradycardia lura a lokacin lokaci daya gwamnati na magani don magunguna "trimetafan", "mecamylamine", "guanadrel", "guanethidine." Kara gida m ayyuka tara kudi "Epinephrine," "methoxamine", "Phenylephrine."

Features na aikace-aikace

Kafin tsarma "Novocaine" da kuma yin harbi, ake bukata dole domin sanin mutum ji na ƙwarai to magunguna. Don yin wannan, gudanar da wani fata gwajin, kuma idan akwai redness da kuma kumburi za a iya hukunci a kan wani mutum ba yarda nufi.

A lokacin jiyya da shi wajibi ne don saka idanu aiki na zuciya da jijiyoyin jini, juyayi da kuma numfashi tsarin. Don rage na tsari mai daukan hotuna, yawan guba da kuma kara da sakamako daga cikin miyagun ƙwayoyi a lokacin da maganin sa barci, da miyagun kwayoyi "lidocaine" ko "Novocaine" da ake amfani a tare da tare da vasoconstrictors. Domin wannan, daya drop of epinephrine hydrochloride bayani da aka kara to 3 ml na medicament "Novocaine".

A mafi girma da taro na bayani amfani, da karin ne mai guba miyagun ƙwayoyi. Don rage tasiri dakarun shi bada shawarar rage overall sashi na medicament ko diluted zuwa ƙananan taro. Wannan ne yake aikata tare da wani bakararre isotonic bayani na sodium chloride.

Domin rigakafin wani hypersensitivity dauki a matakin farko na lura gudanar 2 ml biyu-kashi bayani, da kuma bayan kwanaki uku (idan babu illa) da kashi da aka karu zuwa 3 ml, sa'an nan fitowa don amfani da cikakken ƙarfi - 5 ml da allura.

A lokacin outpatient magani ake bukata ba up tuki da kuma aiwatar da ayyuka alaka da ƙãra da hankali, gudun mota da hankulansu halayen.

Hulda da sauran kwayoyi

Lokacin gudanar intravenously, da miyagun ƙwayoyi kara habaka hana ruwa guda sakamako a kan m tsarin sedatives, kwayoyin maganin barci, kayayyakin amfani ga babban maganin sa barci, tranquilizers da narcotic analgesics. Da miyagun ƙwayoyi prolongs da mataki na tsoka, jijiya block lalacewa ta hanyar suxamethonium. A hadarin hypotension an karu da hade da yin amfani da kudi "Novocaine" da Mao hanawa).

Anticholinesterase kwayoyi kara da yawan guba daga cikin miyagun ƙwayoyi, hana ta hydrolysis. Para-aminobenzoic acid, wanda shi ne mai metabolite da miyagun ƙwayoyi, rage-rage antimicrobial sakamako na sulfonamides, saboda sun yarda m antagonist. Yiwuwar gida halayen a cikin nau'i na edema, kuma Ya ƙãra wajen kisa a cikin aiki da sarari injections na gida m gwamnati via disinfectant mafita dauke da nauyi karafa.

Da amfani da "Novocaine" miyagun ƙwayoyi a lokacin daukar ciki

A lokacin haihuwa da yawa mata suna fuskantar tare da bukatar hakori magani ko daban-daban m cututtuka, kamar ciwon baya. A Dentistry, maganin sa barci da ake amfani da mafi sau da yawa yana nufin "Novocaine". Amfani da miyagun ƙwayoyi a cikin wadannan yanayi ne m. Ka kawai bukatar sanar da likita game da ciki da cewa ya yi amfani da miyagun ƙwayoyi, shan la'akari da halin da ake ciki. Lokacin da toxicosis, a ci gaba da canji a cikin jini, kamar yadda halatta magani "Novocaine". A ciki, ta yin amfani da mai yiwuwa ne kawai a dagagge matsa lamba, bayan kafin tare da shawara da likita.

Tool facilitates aikin na zuciya da kuma shakatawa sakamako a kan tsokoki. Lokacin da ãyõyin jin zafi a ciki, wanda suna hade da peptic miki cutar, mu bayar da shawarar yin amfani da suppositories. Maido matsa lamba basur ma zai yiwu ta amfani da suppositories. Drug "Novocaine" da aka yi amfani da lokacin daukar ciki ne kawai a kan takardar sayen magani, kai-magani ba a halatta! A gwani zai lissafi da ake bukata kashi da kuma mita na gwamnati, bayan nazarin da Manuniya ciki. Suppositories ana amfani da kullum sau biyu, pre-share jiki via enema.

Price da miyagun ƙwayoyi analogues "Novocaine"

Cost "Novocaine" shiri (price iya bambanta dan kadan a cikin mutum Pharmacy) a vials (0.5%) ne 22 rubles. Per vial 0.25% bayani (200 ml) ko rectal suppositories zai ba 27 rubles. Tsarin analogues na aiki abu ne medicaments:

  • "Procaine hydrochloride".
  • "Novocain tushe."
  • "Novocaine-vial".
  • "Novocaine Bufus".

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