"Sumatriptan": umarnin don amfani, reviews. Drug analogues "Sumatriptan"

Abin da ake nufi da miyagun ƙwayoyi "Sumatriptan"? Umurnai na yin amfani da miyagun ƙwayoyi, da pharmacological mataki, da kuma tsari na abun da ke ciki za a gabatar kadan kara. Har ila yau, a wannan labarin, za mu gaya muku game da abin da Contra-alamomi da kuma gefen sakamakon wannan magani yana da, abin da hanyoyin da aikace-aikace da kuma sashi, idan ya na da wani analogues da sauransu.

A abun da ke ciki na magani da kuma abun da ke ciki

A halin yanzu, kawai kwayoyi za a iya samu a Pharmacy da hanci fesa "Sumatriptan". Umurnai na yin amfani da wannan kayan aiki na samar da cikakken bayani a kan abun da ke ciki na miyagun ƙwayoyi. Saba da shi za ku iya zuwa yanzu.

A fim mai rufi Allunan dauke da aiki abu kamar sumatriptan succinate. Game da karin abubuwa, wadannan sun hada da wadannan: alli hydrogen phosphate dihydrate, microcrystalline cellulose, giproloza (Klutsel ko hydroxypropylcellulose LF), magnesium stearate, mannitol (ko mannitol), croscarmellose sodium (ko primelloza).

The aiki sashi hanci fesa "Sumatriptan" kuma hidima sumatriptan. Amma ga karin aka gyara, su za a iya canja bisa ga siffar da medicament saki. Ya kamata a lura da cewa SPRAY da aka amfani da su bi nisa ƙasa da na kowa, fiye da Allunan. Duk da haka, suna da nasu masu amfani. Matsayin mai mulkin, waɗannan su ne marasa lafiya da suke ba dadi shan magani da baki.

A pharmacological halaye na da miyagun ƙwayoyi

Abin da siffofin ne "Sumatriptan" Allunan, wanda sake bitar mu duba kara?

Ya ce shiri ne a protivomigrenoznoe nufi. Yana da wani takamaiman da zabe agonist na 5-HT1-serotonin rabe, wanda ake sarrafa a cikin jini da finjãlai na kwakwalwa. Ya kamata a lura cewa da miyagun ƙwayoyi yana da wani sakamako a kan sauran subtypes na 5-HT-serotonin rabe.

Bayan shan miyagun ƙwayoyi shi sa vasoconstriction na carotid jijiya gado. Saboda haka, medicament "sumatriptan" (Allunan) SUPPLiES jini intracranial da extracranial kyallen takarda. Ya kamata a lura da cewa shi meningeal vasodilatation, kuma su kumburi da suke haddasawa migraine a cikin mutane.

Ba za mu iya ce cewa bayan da tallafi na kayan aiki da wannan yana da wani gagarumin sakamako (korau) a kan cerebral jini ya kwarara. Allunan kawai hana tsoka mai amsa sigina aiki na afferent zaruruwa (su endings) na trigeminal jijiya, wanda aka located a cikin Dura. Wannan na faruwa saboda da rage na azanci shine neuropeptide saki.

Ya kamata kuma a ce cewa miyagun ƙwayoyi "Sumatriptan" da "Sumatriptan Teva" gaba daya kashe photophobia da tashin zuciya, wanda aka kai tsaye nasaba da migraine harin.

A tasiri daga cikin miyagun ƙwayoyi

Ta yaya sauri zo da kyau sakamako bayan da tallafi na "Sumatriptan" miyagun ƙwayoyi? Shedu wannan medicament dauke da bayanai da cewa da miyagun ƙwayoyi fara aiki ne kawai bayan minti 30. Kamar wancan ne da haƙuri ya riƙi wani kashi na 100 MG. Ba zato ba tsammani, a 50-70% da marasa lafiya da sauri suna shafe migraine hare-haren bayan yin amfani da 25-100 MG na da miyagun ƙwayoyi. A lokacin da rana a 1/3 marasa lafiya da komowa, wanda ke bukatar maimaita yin amfani da miyagun ƙwayoyi.

Pharmacokinetics

miyagun ƙwayoyi "Sumatriptan" Har yaushe tunawa? Amsar wannan tambaya kuma an samu a cikin umarnin don yin amfani da kudi. Bayan karbar magani a ciki, ya kusan nan da nan tunawa a cikin narkewa kamar fili. Bayan game da minti 45 da taro na miyagun ƙwayoyi a cikin jini magani kai game da 70%.

Saboda bai cika sha da farko-izinin metabolism, da cikakkar bioavailability da miyagun ƙwayoyi a lokacin gudanar a kan talakawan 14%. Game dauri ga jini jini sunadarai, yana da matukar low (game da 15-21%). A rabin-rai lokaci ne game da 2-hours. Shiri samu yawanci ta hanyar da kodan.

Absorbability da miyagun ƙwayoyi a takamaiman asibiti yanayi

Bisa ga art, migraine kai hare-hare ba muhimmanci shafar absorbability na aiki wakili sumatriptan (by ingestion ko intranasal gwamnati).

Idan haƙuri ne gaji da damuwa da hanta aiki, sa'an nan bayan yin amfani da magani ya iya samun wani ƙara matakin na aiki sashi a cikin jini. Wannan na faruwa a sakamakon rage farko-izinin yarda.

Alamomi ga yin amfani da magunguna

A wasu lokuta, prescribers "Sumatriptan"? Umurnai na yin amfani da miyagun ƙwayoyi ce cewa ya kamata a dauka kawai tare da manifestations na migraine (ba tare da Aura ko ta).

Contraindications ga yin amfani da

Idan akwai sabawa shi ne tsananin haramta dauki magani "Sumatriptan" analogs wannan magani? Ina so in jaddada cewa, a wannan batun a cikin umarnin akwai babban adadin bayanai. Wannan shi ne dalilin da ya sa kafin shan miyagun ƙwayoyi da shi, tabbata a karanta.

To, abin da suke da Contra-alamomi ya nuna da miyagun ƙwayoyi? Ka yi la'akari da jerin yanzu:

• ƙara ji na ƙwarai daga mãsu haƙuri ga abubuwa na halitta.
• Tsofaffi da marasa lafiya (a kan shekaru 65);
• basilar, ko oftalmoplegicheskaya form hemiplegic migraine.
• lokaci daya liyafar da wani medicament da medicaments wanda dauke da ergotamine da daban-daban Kalam, kazalika da Mao hanawa (haramta daga karbar nufin kafin kwanaki 14 bayan janyewar ce kwayoyi).
• jijiyoyin zuciya da cututtukan zuciya, da kuma da ake zargi da shi.
• matashi da yara shekaru (18 years).
• angina, ciki har da Prinzmetal angina .
• ciki da kuma nono.
• tsokar zuciya infarction, ciki har da gudãna a cikin tarihi.
• hauhawar jini (uncontrolled irin).
• hauhawar jini (sarrafawa irin).
• occlusive na gefe jijiya cuta.
• epilepsy, ciki har da wani pathological yanayi hade tare da low farfadiya ƙofa.
• koda ko hanta gazawar;
• bugun jini ko dõgẽwa Jihar cerebral jini ya kwarara, ciki har da kwarara tarihi.

Kamar yadda aka ambata a sama, da miyagun ƙwayoyi "Sumatriptan" dole ne ba a yi amfani da lokacin daukar ciki. Amma idan hadarin da tayin ne kasa da amfani zuwa ga uwar, shi ne har yanzu wajabta mata a jihar da kuma masu jego. Duk da haka, ka yi wannan ne don kawai wani gogaggen gwani (da miyagun ƙwayoyi ne riƙi tsananin karkashin ta dubawa). Af, shi ba da shawarar don ciyar da jariri da nono cikin wani yini bayan samun ce Allunan.

Drug "Sumatriptan": umarnin don amfani da

Wannan magani an dauka baki, ko da kuwa abinci ci. Sashi a cikin wannan harka dole ne daidai da 50 MG (idan da ake bukata - 100 MG).

Idan ka shawarta zaka tambaya hanci medicament "Sumatriptan" (fesa), ta kashi ne 20 MG a kowane ƙofar hanci. Maimaita gwamnati da miyagun ƙwayoyi ne a yarda ba a baya fiye da bayan 2 hr.

A kalla kullum sashi na baka gwamnati ne 300 MG. Lokacin amfani intranasal halitta, shi ne daidaita biyu allurai 20 MG.

Features magani

Yanzu da ka san yadda za ka lashe a migraine. "Sumatriptan" (Allunan, kuma ya fesa) copes da kyau tare da aiki. Duk da haka, ya kamata a lura da cewa medicament ba a yi nufin ga prophylaxis na ce karkacewa.

Amfani da miyagun ƙwayoyi ne zai yiwu ne kawai a cikin akwati inda ganewar asali ne a cikin shakka. Kafin nadin da miyagun ƙwayoyi "Sumatriptan" marasa lafiya da atypical kuma ba a baya kamu da migraine, likita dole ne su tabbatar da sarauta daga sauran neurological yanayi m. Ya kamata kuma a haifa tuna cewa marasa lafiya da ganewar asali bayan da tallafi na ce Allunan iya ci gaba cerebrovascular cuta.

A gaban munanan a cikin jijiyoyi (a cikin maza girmi 40 shekaru da kuma postmenopausal mata) na bukatar wani na farko jarrabawa domin ware munanan na zuciya da jini.

A halin yanzu akwai bayani game da abin da ya faru na take hakki da daidaituwa, wani rauni da hyperreflexia bayan shan miyagun ƙwayoyi, "Sumatriptan" da sauran kwayoyi daga cikin rukuni na zabe mai hanawa.

Kafin da kuma a lokacin jiyya da miyagun ƙwayoyi gabatar na bukatar m abinci ci, kazalika da riko da wani m rage cin abinci. Saboda haka, haƙuri kamata kashe daga abinci da abinci ke dauke da tyramine abu (cakulan, Citrus, koko, seleri, kwayoyi, cuku, wake, da kuma tumatir). Bugu da kari, wajibi ne ta yi watsi da amfani da giya, ciki har da ja, kyalkyali da kuma bushe giya, shampen, giya.

Motsa jiki da kuma rike da lafiya salon a general (na tafiya, iyo, gudun kan), kazalika da gaban wani sha'awa taimako zuwa fitowan tabbatacce motsin zuciyarmu, wanda ya hana ci gaban wani mutum haƙuri na migraine harin.

Umarnin a kan yin amfani da wani hanci SPRAY

Ciniki sunan fesa tare da aiki abu sumatriptan sauti kamar "Imigran". Wannan magani yana da wadannan sassa:

• matsa yatsunsu.
• wani tip.
• blue wani button.

Ya kamata a lura da cewa blue button da aka kunna sosai da sauri da kuma sau ɗaya kawai. A wannan dangane shi ne shawarar ba ka danna a kan shi, har tip aka shiga hanci nassi. In ba haka ba, da cikakken kashi za a tafi a banza.

Don amfani da hanci SPRAY, da mãsu haƙuri ya riƙi wani wuri dadi, kwance, ko a tsaye da zaune. Af, bayan da mãsu haƙuri ta hanci kogo bada shawarar da za a tsabtace tare da auduga swabs.

Ana cire da bororo fakitin kuma cire da miyagun ƙwayoyi domin hanci amfani, da miyagun ƙwayoyi dole ne a shiga cikin daya ƙofar hanci. Amma ga sauran hanci nassi, dole ne a guga man a yatsa ga hanci septum. A wannan yanayin, da mãsu haƙuri dole ne numfashi ta bakin.

Saka tip cikin ƙofar hanci hanci halitta ya zama 1 santimita. The shugaban na haƙuri kamata ci gaba mike, ba jefa baya baya. Bayan haka, haƙuri kamata rufe bakinsa da kuma yin shiru da kuma jinkirin breaths ta hanci, tare da wani lokaci daya kokarin danna kan blue button tare da yatsa. A wannan yanayin, wani mutum zai iya ze cewa button ne sosai m. Amma wannan ba shine al'amarin ba. A lokacin da allura daga cikin miyagun ƙwayoyi a cikin hanci rami na haƙuri kamata ji wani suma danna sauti. Wannan yana nufin cewa button ya samu nasarar aiki.

Bayan wannan hanya, da mãsu haƙuri ake bukata don bude bakinsa da kuma numfashi sannu a hankali ta hanyar da shi. Head dole ne ci gaba da kiyaye madaidaiciya. Next, da mãsu haƙuri ya kamata su sa a shiru numfashin ta hanyar hanci kogo, da kuma for sa'an nan exhale - ta bakin (for 10-20 seconds). An shawarar ba numfashi ma warai.

Da zarar an kammala hanya da allura daga cikin miyagun ƙwayoyi, mutum zai iya ji gaban danshi a cikin hanci, kuma matalauta iyawa. Wadannan majiyai ba kawo hadari ga kiwon lafiya da kuma sauri wuce spontaneously. Bayan guda aikace-aikace na jin za a iya jefar da.

Tsõratar da lokacin da yin amfani da

Drug "Sumatriptan Teva", reviews daga waxanda suke da kyau zuwa mafi girma har, shi ya kamata a dauka tare da matsananci hankali ga direbobin motocin, kazalika da waɗanda suka tsunduma a m ayyuka da cewa bukatar ƙara rates na dauki da kuma hankali.

illa

Iya tsokana gefen sakamakon da magani "Sumatriptan"? Shirye-shirye na wannan irin na iya taimakawa ga ci gaban da wani fairly manyan yawan korau mamaki. Bari mu bincika su, a cikin mafi daki-daki:

• mutum jijiyoyi. A wani ɓangare na tsarin a cikin wani haƙuri low jini iya lura, tsokar zuciya infarction, dan lokaci hawan jini (yawanci jim kadan bayan ingestion), tachycardia, bradycardia, tachycardia, da kuma a wasu lokuta, arrhythmia, spasms da jijiyoyin zuciya arteries, mai shudewa ECG canje-canje Raynaud ta ciwo.
• Juyayi tsarin da kuma ji gabobin. Bayan shan miyagun ƙwayoyi da mutum zai iya fuskanci gajiya, juwa ko jiri, wani rauni da drowsiness. A wasu lokuta, da miyagun ƙwayoyi sa diplopia, seizures, da ya faru na flicker kwari kafin idanunsa, nystagmus, rage gani acuity, scotoma kuma m mai shudewa asarar hangen nesa.
• Narkewa kamar fili. Daga cikin narkewa a cikin haƙuri sau da yawa gani amai, dysphagia, tashin zuciya, da kuma kara (qananan) aiki na hanta enzymes, na ciki da rashin jin daɗi da kuma ischemic colitis.
• Alerji. Bayan shan miyagun ƙwayoyi, da wasu marasa lafiya ruwaito bayyanar pruritus, rash, urticaria da erythema. Har ila yau, akwai anaphylaxis, jin zafi, tingling da kuma zafi a kai, wani nauyi, matsa lamba, flushing, kuma myalgia. Intranasal gwamnati da miyagun ƙwayoyi iya faruwa a cikin nau'i na gida halayen huhu dõgẽwa hangula ko kona abin mamaki a cikin makogwaro da karan hanci kogo da kuma hanci zub da jini.

Hulda da sauran kwayoyi

Yaya sauran magunguna a kan tasiri da kuma tasirin da "Sumatriptan" miyagun ƙwayoyi? Umurnai, comments daga masana a kan wannan batu dauke da wadannan bayanai. Tare da lokaci daya da yin amfani da miyagun ƙwayoyi da medicament "Ergotamine" kuma na nufin wani haƙuri ergotaminsoderzhaschimi yiwu dogon vasospasm. A wannan batun, da tazara tsakanin allurai da wadannan kwayoyi ya kamata a kalla 24 hours.

Bisa ga binciken, akwai wani hulda tsakanin miyagun ƙwayoyi "sumatriptan" da kuma Mao hanawa. Kamar wancan ne da rayuwa kudi an rage farko, kuma ta maida hankali ƙaruwa.

Tare da lokaci daya amfani da ce anti-migraine kwayoyi, da kuma mallakar zabe serotonin reuptake hanawa, da mãsu haƙuri iya ci gaba da rauni, hyperreflexia kuma gaji da damuwa da daidaituwa na ƙungiyoyi.

Yawan abin sama da kwayoyi (bayyanar cututtuka, magani)

Me zai faru idan ba ka bi da sashi shawarar da likita? Lokacin da ya wuce kima yin amfani da shiri "sumatriptan" marasa lafiya na iya kara sama gefen halayen. A wannan batun, hãlãyensu bukatar musamman kallo don 10 hours.

Idan dole, wani yawan abin sama haƙuri ne taimaka a cikin nau'i na symptomatic magani.

Drug "Sumatriptan": analogues da miyagun ƙwayoyi farashin

Saya da kayan aiki a wani kantin magani. Ya kamata a lura cewa farashin "Sumatriptan" da miyagun ƙwayoyi, idan aka kwatanta da sauran, in mun gwada low. Saboda haka, a kan 50 film mai rufi alluna za ka biya kawai 170-200 Rasha rubles. Amma ga hanci yana nufin cewa da price ne game da wannan.

ko takwarorinsu da miyagun ƙwayoyi "Sumatriptan"? "Amigrenin" - wani magani da aka fi samu kawar da migraine kai hare-hare idan sama yana nufin ba ya nan daga cikin kantin magani. Bayan shi, analogues medicament "sumatriptan" na aiki abu ne da wadannan kwayoyi: "Sumarin" "Imigran", "Sumitran", "Migrepam", "Sumatriptan-Teva", "sumatriptan succinate", "sumatriptan Pfizer", "sumatriptan Adifarm "" Sumamigren "," Trimigren "da sauransu.

Har ila yau, kamar yadda mai kama da hanci decongestants, wasu masana bayar da shawarar yin amfani da SPRAY "Imigran".

Storage yanayi da kuma shiryayye rai

Gabatar miyagun ƙwayoyi ya kamata a adana kawai a bushe kuma kariya daga hasken rana wuri. A zafin jiki a cikin dakin kada ta kasance fiye da 25 digiri. A shiryayye rayuwar likita da wuraren ne shekaru 3. Bayan wannan lokaci, da miyagun ƙwayoyi dole ba za a yi amfani da.