Kiwon lafiyaShirye-shirye

Umarnin don amfani "tiapridal". Analogs da kuma sake dubawa

"Tiapridal" - antipsychotic magani kerarre da tiapride. Da miyagun ƙwayoyi ne amfani a matsayin magani mai kantad da hankali, analgesic da kuma hypnotic. Dalili na antipsychotic mataki - tarewa da dopamine rabe, wanda muhimmanci shafi aiki na CNS. A wannan labarin, za mu bayyana a cikin daki-daki, game da miyagun ƙwayoyi.

Abun da ke ciki hada da miyagun ƙwayoyi

A magani yana samuwa a cikin biyu siffofin, da kwamfutar hannu za a iya saya, kuma da bayani:

  • Daya kwamfutar hannu kamar yadda daya ampoule qunshi 100 milligrams na babban bangaren da karin abubuwa. Kamar yadda karin sinadaran amfani da abun da ke ciki na povidone, magnesium stearate, mannitol. A abun da ke ciki ne kuma suna goyon bayan da wani mai ruwa-ruwa colloidal dioxide, silicon da microcrystalline cellulose.
  • Baya daga cikin babban bangare ne na bayani qunshi sodium chloride da ruwa ga allura.

A daya akwatin dauke 20 Allunan (2 blisters da 10 Allunan) ko 12 vials (2 blisters na 6 vials). Umarnin don amfani "Tiapridal" a cikin nau'i na wani bayani ga allura damar gudanar intravenously da intramuscularly. Wannan nau'i na da miyagun ƙwayoyi ne kawai dace domin lura da adult marasa lafiya.

Pharmacodynamics "tiapridal"

A medicament yana neuroleptic, analgesic da anxiolytic mataki. Kamar yadda umurci manual, "Tiapridal" selectively tubalan aiki na D 2 rabe na tsakiyar dopamine. Kamar wancan ne a kan D 1 rabe yana da wani sakamako. Da miyagun ƙwayoyi samun kawar da psoriasis, a lokacin da amfani a cikin tsofaffi inganta tunanin.

Pharmacokinetics "tiapridal"

Intramuscular gwamnati da miyagun ƙwayoyi (200 MG) na matsakaicin matakin a cikin jiki da aka gano bayan minti 30, ta amfani da Allunan, a wannan kashi - 60 minutes. A bioavailability da miyagun ƙwayoyi a lokacin da amfani da nan da nan kafin abinci tare da 75% ya karu zuwa 95%. Saboda kwayoyi irin amfani ƙaruwa da matsakaicin matakin a wani kwayoyin (40%).

Absorption a cikin jiki ne hankali a tsofaffi da marasa lafiya. "Tiapridal" umarnin don amfani na nufin wani wakili crosses da placental da jini-kwakwalwa shinge. An sani cewa a lokacin jiyya da miyagun ƙwayoyi ne ba a cikin abun da ke ciki na nono madara. A mata, da m kau da miyagun ƙwayoyi da sauri fiye da na maza (a kan 2.9 hours), bambanci ne 0.7 hours. Metabolism halin a matsayin matsakaici. Babban ɓangare na miyagun ƙwayoyi (70%) an cire daga jiki da kodan canzawa.

Alamomi "Tiapridal" shirye-shiryen

Don aiwatar da far da kwayoyi "Tiapridal" karatu kamar haka:

  • dyskinesia (tardive, maras wata-wata).
  • Gilles de la Tourette ciwo.
  • chorea.
  • halayya cuta (m jihar, agitation et al.), sakamakon wani gwaji da kwarara na kullum shan barasa da kuma tsofaffi da marasa lafiya.
  • korau bayyananen a hali, kamar m jihar da kuma agitation.
  • zafi m hali (na kullum form).

Contraindications, gazawar zuwa sama "Tiapridal" miyagun ƙwayoyi

Ya haramta Kaddamar da "Tiapridal" umarnin don yin amfani da yara wanda shekaru ne kasa da shekaru shida. A na yara far ne da za'ayi kawai kwayoyi. A miyagun ƙwayoyi ya kamata ba a bi da mata masu juna biyu da kuma marasa lafiya da suke nono. Magani da ba a amfani a yanayin saukan hypersensitivity to da aka gyara, da sauran irin wannan wajen. Contraindications hada da irin jihohi:

  • hanta da na koda gazawar, wanda yana da babba mai tsanani.
  • prolaktinzavisimogo diagnosing marurai, zargin da ta hallara.
  • hawan jinni rikicin.
  • ganewar asali pheochromocytoma, a tuhuma da ta zama.

Allunan, kuma da bayani da ake amfani da tare da "sultopride" da kuma dopamine tsoka mai amsa sigina agonists (da togiya ne lura da marasa lafiya da Parkinson ta cuta) ba a hade tare da wasu iri neuroleptics, anti-arrhythmic jamiái na zuwa azuzuwan Na kuma III A.

Medicating "Tiapridal" wa'azi ba da damar a lokaci guda ta amfani da "Moxifloxacin", "sparfloxacin", "Difemanila", "Erythromycin", "bepridil," "mizolastine", "levodopa", "cisapride" kuma tare da igiyar jini "vincamine" .

Idan haƙuri (musamman tsofaffi) ana bi da tare da kwayoyi da cewa zai iya kai wa ga ci gaban hypokalemia, cardiac madugu tabarbarewar, tsawon kwanakinka QT tazara, da ya faru na bradycardia bayyana hali, amfani da "Tiapridal" dole ne a hankali. Tsanaki ake bukata a cikin irin wannan hali:

  • Parkinson ta cutar.
  • nakasar QT tazara elongation hali.
  • hypokalemia.
  • kullum na koda gazawar.
  • bradycardia.
  • cututtuka a wadda lalace zuciya da jijiyoyin jini tsarin (decompensation mataki).
  • epilepsy.

Jiyya tare da "Tiapridal"

a kan aikace-aikace na "Tiapridal" manual ya bayar da shawarar yin amfani da wata na farko a cikin kananan allurai, a hankali kara su, domin ya sami matsakaicin sakamako.

halayya cuta

Domin su taimako wajibi ne a yi amfani da 200 MG na da miyagun ƙwayoyi kullum (har zuwa 300). A tabbatacce sakamako aka samu a makonni shida a kan talakawan. Mazan marasa lafiya gudanar da wani m kashi na magani - 50 MG. A guda kashi kamata a cinye sau biyu a rana, da kuma ta karuwa yake halatta a yarda da kayyade tazara, da mataki da aka yi a hankali, shan la'akari gwani shawara. A kullum kashi kada wuce 300 MG.

Kullum m zafi

A kullum kashi na magani domin lura da irin wannan yanayin ne daga 200 zuwa 400 MG.

Chorea, Gilles de la Tourette ciwo

Lokacin dauke da fitar da magani daga yaro kullum kashi da aka zaba shan la'akari da jiki nauyi da kuma game da 3-6 MG / kg. Idan kana bukatar ka gudanar da wani adult far, da farko yi amfani da 25 MG da miyagun ƙwayoyi a kowace rana, daga baya (bayan wani sauka a hankali karuwa a kashi) - 300-800 MG.

Agitation, ta'adi

The shawarar kullum kashi na medicament ne daga 100 zuwa 150 MG.

halayya cuta

The shawarar kashi na rana amfani (daga 200 zuwa 300 MG) a yanayin saukan delirious jihohi ko predelirioznogo yakan to 400-1200 MG. Matsakaicin yiwu kashi wanda dole ba za a wuce, shi ne 1800 MG. A gabatarwar da miyagun ƙwayoyi samar a kan talakawan kowane sa'o'i biyar. Idan magani wajibi ne ga tsofaffi mutum, a kowace rana shi ne 2-3 injections tsakanin wanda ya lura tazara na 6 hours. Domin lura da irin marasa lafiya shawarar kullum ci daga 200 zuwa 300 MG na medicament a lokaci da aka yarda su shigar da kasa da 100 MG "tiapridal".

M magana da wani kullum yanayin zafi

Hanyoyin kwantar da hankali dangane da gudanar da kullum kashi m zuwa 200-400 MG na da miyagun ƙwayoyi.

Side effects lokacin shan "Tiapridal" miyagun ƙwayoyi

Lokacin zalunta miyagun ƙwayoyi "Tiapridal" umurci manual, reviews tabbatar da alama na wasu m halayen. Take hakkin iya faruwa a cikin urogenital, juyayi, endocrine da zuciya da jijiyoyin jini tsarin. Bugu da kari, akwai wani hadarin matsalolin da hankula. Ga wasu illar hada da allergies, fata bayyananen tare da nauyi riba, orthostatic hypotension.

Yawan abin sama "tiapridal"

Idan ka yi amfani da} arfin kashi yiwu yawan abin sama da kuma ta bayyanar cututtuka sun hada da disturbances na sani, mafi tsanani daga wanda - coma, neuroleptic ciwo (m, m siffofin). Domin magance wannan jiha da kwayoyin ne da za'ayi magani bisa anticholinergic jamiái. Bayan da yarjejeniyoyin da miyagun ƙwayoyi zama dole don gudanar da wani symptomatic magani da kuma plasmapheresis.

tsõratar

Kafin yin amfani da wani magani "Tiapridal" umurci manual bada shawarar cewa ka gyara hypokalemia. A lokacin far yana da muhimmanci a kullum saka idanu electrolyte balance, gudanar da wani electrocardiogram, saka idanu da na asibiti hoto canje-canje.

Idan ya zama dole a yi amfani anticholinergic kwayoyi haifar samun neuroleptics extrapyramidal ciwo raya maimakon dopamine tsoka mai amsa sigina agonist.

A lokacin magani ya kamata bari ayyuka da cewa gabatar da wani m barazana, shi ba da shawarar yin aiki bukata musamman kula da sauri martani.

Hulda da sauran abubuwa

Wasu hade shirye-shirye tare da shan magani "Tiapridal" wa'azi, feedback hade da yiwuwar faru na undesired halayen. An ba da shawarar a lokacin jiyya da amfani "Clonidine", antihistamines, anxiolytics, barbiturates da opioids, kamar yadda "tiapridal" sakamako zai zama mafi pronounced. Saboda incompatibility ba za a dauka "levodopa" da kuma barasa. Magani za a iya hade tare da yin amfani da neurotrophic kwayoyi, analgesics, antidepressants, neuroleptics. Babban hadarin da orthostatic hypotension, akwai lokaci daya amfani da antihypertensive kwayoyi tare da "Tiapridalom".

A kudin magani analogues, sake bitar game da miyagun ƙwayoyi "Tiapridal"

Idan dole magani "Tiapridal" yana nufin koyar da bayanin bari ka san abin da wani magani ne. A farashin da kwayoyi ne na bayar da muhimmanci a zabin da wani medicament domin magani. The bayani a vials za a iya sayi for game da 995 rubles, da Allunan - for 1,400 rubles.

Daga cikin analogues da miyagun ƙwayoyi - "Eglonil", "Betamax". Na musanya iya zaba "Sulpiride" ko "Prosulpin". Akwai wani analogue da miyagun ƙwayoyi - "tiaprid", ya ke dauke da mafi m, shi ne quite wani mashahuri wani zaɓi, da m miyagun ƙwayoyi samarwa wanda ke hulda da kamfanin "Organic". Kamar yadda wani ɓangare na "tiaprid" gabatar da wannan aiki abu, wanda shi ne wani ɓangare na magani "Tiapridal". Anfani analogs Guide bada shawarar a zabi, a lokacin da asali ba za a iya amfani da lokaci guda tare da wasu kwayoyi sa illa da ba samar da wani so sakamako. Don da miyagun ƙwayoyi ya fi tasiri, la'akari da yawa na da maki a lokacin zaɓa.

A lokacin jiyya, yana da muhimmanci a bi duk likita ta da shawara da kuma shawarwari, wanda ya ƙunshi umarnin don amfani. "Tiapridal", kamar yadda aka nuna ta hanyar feedback, a mafi yawan lokuta, da ake amfani da su kawar da yanayi tare da juyayi da tashin hankali da kuma m hali, giya psychosis. Yawancin lokaci, marasa lafiya da likitoci gamsu da sakamakon far. Amma, a refresher shakka ba da ake bukata domin dalilin cewa so sakamako ne masu tasowa, bayan da aiwatar da farko hanya. Reviews nuna cewa ga marasa lafiya magani "Tiapridal" sauki don amfani.

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