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"DITT difo": umarnin don amfani, contraindications, illa, reviews, photos

Me ka sani game da wannan magani, kamar "DITT difo"? Umarnin don amfani, contraindications, reviews da kuma gefen sakamakon da miyagun ƙwayoyi za a yi la'akari da kara.

Marufi da kuma nau'i na da miyagun ƙwayoyi, da abun da ke ciki

A abin da siffar samar da wani magani da "DITT difo"? Umurnai na amfani rahotanni cewa za a iya saya a cikin nau'i na wani m bayani ga intramuscular allura. Babban aiki sashi na wannan miyagun ƙwayoyi ne fluphenazine decanoate. Kamar yadda shi shiga sayar da duhu gilashin ampoules, pre-kunsasshen a cikin cell kwane-kwane da kuma takarda fakitoci, bi da bi.

pharmacology

Mene ne magani Properties muhimmi medicament "DITT difo"? Umurnai na amfani, da sake dubawa ce cewa wannan shi ne wani dogon-aiki antipsychotic magani. A nasa ne a rukuni na polyvalent neuroleptics da kuma farfado furta antipsychotic Properties, wanda ake hada tare da jawo kuma antiemetic sakamako. Har ila yau, wannan magani yana da wani m magani mai kantad da hankali sakamako.

Abin da ya haddasa tasiri na da miyagun ƙwayoyi "DITT difo"? Umurnai na amfani furta cewa, ta antipsychotic effects hade tare da kawancen na dopamine D2 rabe Mesocortical da mesolimbic tsarin.

Magani mai kantad da hankali Properties na wannan medicament da moderately bayyana ne kawai a lokacin da ya lura high allurai na bayani. Su ne saboda kawancen na adrenergic rabe na mutum sassan na kwakwalwa kara.

Game da anti-emetic effects na magani, to, shi ake dangantawa da kawancen na dopamine D2 tsoka mai amsa sigina jawo sashi daga cikin amai cibiyar. Ya kamata kuma a lura da cewa hypothermic sakamako na wannan magani ya nuna kawancen na dopamine rabe na hypothalamus.

Ta yaya da yawa miyagun ƙwayoyi fara aiki "DITT difo"? Umurnai na amfani (photo allura bayani gabatar a cikin wannan takarda) rahoton cewa warkewa sakamako daga cikin miyagun ƙwayoyi ne yawanci bayyana bayan 25-72 sa'o'i bayan da allura. Ya kamata kuma a lura cewa da kaddarorin na antipsychotic miyagun ƙwayoyi a karkashin shawara suna mafi furta a lokacin daga 49 zuwa 97 hours bayan gwamnati na bayani.

A motsi da miyagun ƙwayoyi

Mene ne halayyar da pharmacokinetics da miyagun ƙwayoyi "DITT difo"? Umurnai na yin amfani da da'awar cewa fluphenazine a cikin nau'i na high kwayoyin nauyi ester mai bayani daga m acid zai iya tara a adipose depots, kazalika da sannu a hankali saki.

Bayan intramuscular allura a kalla taro na kashi ne samu bayan 25 hours a jini. A wannan yanayin, fluphenazine ta ɗaure to jinin samar da 90%.

An fito da miyagun ƙwayoyi readily crosses da placental shãmaki, kuma ya wuce ta jini-kwakwalwa, da kuma ba su excreted da hemodialysis.

Fluphenazine gaba daya da kuma baje metabolised da hanta enzyme tsarin shafe cytochrome P450. Daga cikin jiki shi ne excreted da bile da fitsari. Active metabolites wannan kashi ne ba cikakken gane.

Fluphenazine rabin rayuwa ne 7-10 hours.

shaidar

A wasu lokuta, da haƙuri da aka wajabta injections "DITT difo"? Umurnai na amfani yana nufin irin wannan shaidar kamar:

  • exacerbation na schizophrenia (for rigakafin).
  • shafe tsawon goyon baya lura da kullum schizophrenia.

Haramta yin amfani da

An fito da magani da aka haramta a cikin wadannan lokuta:

  • karkashin nauyi SS cututtuka, ciki har da tare da decompensated kullum Sistem gazawar da kuma hypotension.
  • a wani dagagge ji na ƙwarai daga mãsu haƙuri ga fluphenazine, kazalika da sauran abubuwa na miyagun ƙwayoyi.
  • zalunta a lokacin CNS da comatose jihohi.
  • a lokacin daukar ciki.
  • a kwanyar rauni, kuma m tsari cututtuka na kwakwalwa da kuma laka.
  • a ciyar;
  • tare da sosai hanta aiki da jini tsarin.
  • har zuwa shekaru 12.

Hankali yin amfani da kwayoyi

Zama wary "DITT difo 'miyagun ƙwayoyi wajabta:

  • shan barasa, kazalika ya karu laulayi hepatotoxic halayen.
  • pathological canje-canje a cikin jini, kazalika a take hakkin hematopoiesis.
  • allergies phenothiazines, ciki har da wani tarihi.
  • ƙulli glaucoma.
  • nono.
  • hanta da kuma / ko na koda gazawar.
  • ulcers na narkewa kamar fili, ciki har da tsawon m rashin lafiya.
  • prostatic hyperplasia da na asibiti manifestations.
  • myxedema.
  • ailments, tare da thromboembolic rikitarwa.
  • Parkinson ta cutar.
  • kullum cutar da numfashi gazawar (ciki har da yara).
  • Reye ta ciwo.
  • epilepsy, amai, seizures.
  • cachexia.
  • a cikin tsufa.

Da miyagun ƙwayoyi bayani "DITT difo": umarnin don amfani da

A ampoules wannan magani ne aka yi nufi ga dogon lokacin da darussa na far (akalla watanni uku). Ya sa hannu kashi ga mafi yawan marasa lafiya ne 12.5-25 MG. M allurai, kazalika da tazara tsakanin gwamnati da mafita m bisa ga warkewa sakamako.

Jiyya da marasa lafiya da hypersensitivity zuwa phenothiazines ya kamata a fara sosai matsa a hankali.

Tsofaffi bukatar nada ƙananan allurai fiye da matasa marasa lafiya (kamar 1/4 to 1/3 na dosing). A wannan yanayin bãyansu bukatar m dubawa.

Mamaki da-hali

Da miyagun ƙwayoyi bayani "DITT difo" na iya haifar da wadannan a ke so dauki:

  • extrapyramidal ciwo, akathisia, tardive dyskinesia, dystopia, oculogyric crises, hyperreflexia, opisthotonos.

  • neuroleptic m ciwo, wanda za a iya m.
  • orthostatic hypotension, sweating, jini da hawa da sauka, tashin zuciya, hypotension, asarar ci, glaucoma, wuce kima salivation, atony mafitsara, polyuria, hanji toshewa, bushe baki, tachycardia, ciwon kai, Heart hangen nesa, maƙarƙashiya, hanci cunkoso.
  • na ramin zuciya arrhythmias, kwatsam mutuwa, na ramin zuciya tachycardia, sakamakon bugun zuciya.
  • mahaukaci lactation, na gefe edema, hailar cuta, hyponatremia, rashin ƙarfi a maza, canje-canje a cikin jiki nauyi, canje-canje a libido a mata;
  • pruritus, exfoliative dermatitis, erythema, seborrhea, urticaria, anaphylactic halayen, photosensitivity, angioedema, Bronchial spasm, laryngeal edema.
  • agranulocytosis, leukopenia, cholestatic jaundice.
  • seizures, zazzabi, ECG canje-canje, babu ja diskinenziyu, amai, venous thromboembolism, lupus-kamar ciwo, da sauransu.

shedu

Yanzu, ka sani, daga abin da ka yi Shots "DITT difo." Umarnin don amfani, illa, kuma contraindications ga yin amfani da wannan bayani ya kuma an tattauna a sama.

Kamar yadda marasa lafiya baya bi da tare da daban-daban antipsychotic kwayoyi, miyagun ƙwayoyi "DITT difo" aiki fiye da nagarta sosai da kuma kawar da duk korau bayyanar cututtuka na schizophrenia. A gabatarwar da wannan miyagun ƙwayoyi ne quite barga kuma dogon lokacin da gafarar.

The kawai drawback na wannan kayan aiki ne da babbar adadin da-hali halayen. A farkon zamanin far a wasu mutane alama hyperthermia, hauhawar jini da kuma autonomic tabarbarewa. Har ila yau, da yawa marasa lafiya da ake gani a giperkinezy tsokoki na baki da kuma fuska, smacked lebe da kuma harshe motsi. Bugu da ƙari kuma, da yin amfani da wannan magani ne sau da yawa ya sa ciki, yana mai sãɓãnin mai tsanani.

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